PROTACS
Physicochemical
properties
workshop
2021
Physicochemical Properties of PROTACS: Challenges and Findings
CASE STUDIES
PROTACS
Physicochemical
Properties
Workshop
2022
SPEAKERS
Mechanistic insight into how PROTACs may cross cell membranes
Jan Kihlberg, Ph.D.
Uppsala University
Designing and optimising PROTACs: Guiding principles and lessons learnt
Alessio Cuilli, Ph.D.
University of Dundee
Optimization of orally bioavailable targeted protein degraders
Brian Cook, Ph.D.
Vividion
Esters vs. Amides: Single-atom substitutions have a big effect on PROTAC properties
Scott Lokey, Ph.D.
University of California Santa Cruz
Lipophilicity beyond octanol/water in the bRo5 chemical space
Giulia Caron, Ph.D.
University of Turin
Discussion Topics
Permeability SAR for PROTACS
In-vitro and in-vivo data correlations
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