Innovative analytical techniques
2021 Physicochemical Properties Workshop
April 1, 2021 @ 1:00pm EST
Physicochemical Properties of PROTACS: Challenges and Findings
Featured Speakers
Mechanistic insight into how PROTACs may cross cell membranes
Jan Kihlberg, Ph.D., Uppsala University
Designing and optimising PROTACs: Guiding principles and lessons learnt
Alessio Cuilli, Ph.D., University of Dundee
Optimization of orally bioavailable targeted protein degraders
Brian Cook, Vividion Therapeutics
Esters vs. Amides: Single-atom substitutions have a big effect on PROTAC properties
Scott Lokey, University of California Santa Cruz
Lipophilicity beyond octanol/water in the bRo5 chemical space
Giulia Caron, University of Torino
Discussion Topics
- Permeability SAR for PROTACS
- In-vitro and in-vivo data correlations
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